Opioides
Tapentadol (Nucynta)
Street names: Nucynta, Palexia, Tapal
Overdose? Act now. Call emergency services — say "unresponsive, not breathing". Give naloxone for opioid-like signs. Hotlines
⚡What it does
- El alivio del dolor de los opioides y la inhibición de la reabsorción de la norepinefrina: el primo más fuerte del tramadol
- Más rápido, más previsible que el tramadol (no hay lotería de CYP2D6)
⚠Key risks
- Calendario II por una razón: perfil completo de adicción a mu-opioides
- Riesgo de convulsiones menor que el tramadol pero presente en dosis altas
- Síndrome de serotonina en combinación
- Retiro de opiáceos estándar - crudo
✚Overdose signs
- Pinpoint pupils
- Slow breathing
- Sedation
Comparación de categoría — Opioides
| Substance | Class | Top risks | Street price |
|---|---|---|---|
| Tapentadol (Nucynta) | Schedule II | Schedule II for a reason: full mu-opioid addiction profile; Seizure risk lower than tramadol but present at high doses | ~$1–$5 per tablet diverted |
| Heroin | Schedule I | Extremely addictive — physical dependence in weeks; Overdose: breathing slows or stops | ~$10–$40 per bag |
| Fentanyl | Schedule II | Respiratory depression; Addiction in days | ~$20–$40 per counterfeit pill |
| Fentanyl HCl (powder) | Schedule II / analogue prosecutions | Lab-purity powder is far stronger than street mixes; Weighing errors are fatal | ~$60–$120/gram wholesale equivalent |
| Acetylfentanyl | Schedule I | ~5–15× weaker than fentanyl but still deadly at gram-level mistakes; Frequent cause of cluster overdoses | ~$25–$60/g where found |
| Furanylfentanyl (Fu-F) | Schedule I | Linked to hundreds of fatal overdoses 2016–2018; Potency similar to fentanyl | ~$20–$50/g |
Street prices are regional estimates. Potency and cuts vary constantly.
?Frequently asked questions
What does Tapentadol (Nucynta) look like?
50–250 mg comprimidos; versiones ER
What are the signs of a Tapentadol (Nucynta) overdose?
Pinpoint pupils; Slow breathing; Sedation Call emergency services immediately and give naloxone if available — it reverses opioid overdoses.
How addictive is it?
Calendario II por una razón: perfil completo de adicción a mu-opioides Dependence can develop with regular use.
🔗Sources & further reading
Facts on this page are compiled from these primary sources. External links open in a new tab.