Performance & Grey-Market Pharma
LGD-4033 (Ligandrol)
Street names: Ligandrol, VK5211, LGD
Overdose? Act now. Call emergency services — say "unresponsive, not breathing". Give naloxone for opioid-like signs. Hotlines
⚡What it does
- SARM — strong muscle-building androgen-receptor agonism
- Human Phase-1 data only (dose-finding for muscle wasting)
⚠Key risks
- #2-selling SARM; case reports of drug-induced liver injury and cholestasis at grey-market doses
- Testosterone suppression stronger than ostarine
- HDL suppression + cardiovascular strain unknown long-term
- Products routinely underdosed, overdosed, or contain different SARMs than labeled
✚Overdose signs
- Jaundice, dark urine (liver)
- Severe lethargy (suppression)
- BP elevation
Category comparison — Performance & Grey-Market Pharma
| Substance | Class | Top risks | Street price |
|---|---|---|---|
| LGD-4033 (Ligandrol) | Not approved; WADA-prohibited; unscheduled | #2-selling SARM; case reports of drug-induced liver injury and cholestasis at grey-market doses; Testosterone suppression stronger than ostarine | ~$40–70 per bottle grey market |
| AICAR (Acadesine) | Unscheduled | No human safety data — cancer-risk flags in cell studies; Sold as research chemical, zero quality control | ~$50–$150 per gram |
| Clenbuterol HCl | Not approved for human use | Racing heart, arrhythmia, tremors; Overdose: dangerous potassium shifts, cardiac events | ~$0.50–$2 per 40 mcg tablet |
| Anastrozole (Arimidex) | Rx-only | Bone density loss, joint pain with long-term use; Crash estrogen too low → depression, libido loss | ~$2–$8 per 1 mg tablet |
| Liraglutide (Saxenda) | Rx-only — not a controlled drug | Sold grey-market at huge markups with counterfeit/refilled pens; Nausea, pancreatitis risk | ~$200–$500 per pen grey-market |
| Naltrexone–Bupropion (Contrave) | Rx-only — not controlled | Bupropion lowers seizure threshold; Misuse for stimulant-like effect is possible but weak | ~$1–$4 per tablet grey-market |
Street prices are regional estimates. Potency and cuts vary constantly.
?Frequently asked questions
What does LGD-4033 (Ligandrol) look like?
Liquid dropper bottles, capsules, raw powder from grey-market peptide/SARM vendors
What are the signs of a LGD-4033 (Ligandrol) overdose?
Jaundice, dark urine (liver); Severe lethargy (suppression); BP elevation Call emergency services immediately.
How addictive is it?
#2-selling SARM; case reports of drug-induced liver injury and cholestasis at grey-market doses Dependence can develop with regular use.